From: Tamoxifen in horses: pharmacokinetics and safety study
Metabolite | |||
---|---|---|---|
4-OH TAM | EDF | N-DMT | |
AUC 0-∞ (pg-mL/min) | 951.1 ± 461.9 | 249.1 ± 238.3 | 131.7 ± 107.6 |
Cmax (pg/mL) | 1.0 ± 0.6 | 0.5 ± 0.4 | 0.2 ± 0.1 |
Tmax (h) | 4.1 ± 4.2 | 3.0 ± 3.5 | 8.0 ± 8.8 |
t1/2E (h) | 9.8 ± 3.7 | ND | ND |